1. ʻO ka sodium Croscarmellose(CMCNa i hoʻopili ʻia): he copolymer i hoʻopili ʻia o CMCNa
Nā Waiwai: Pauka keʻokeʻo a keʻokeʻo paha. Ma muli o ke ʻano i hoʻopili ʻia, ʻaʻole ia e hoʻoheheʻe ʻia i ka wai; pehu koke ia i ka wai a hiki i 4-8 mau manawa o kona nui mua. He wai maikaʻi ka pauka.
Hoʻohana: ʻO ia ka mea hoʻoheheʻe nui i hoʻohana pinepine ʻia. Disintegrant no nā papa waha, nā capsules, nā granules.
2. Kalipuna Carmellose (CMCCa i hoʻopili ʻia):
Nā Waiwai: Pauka keʻokeʻo, ʻala ʻole, hygroscopic. 1% hopena pH 4.5-6. Aneane hiki ʻole ke hoʻoheheʻe ʻia i loko o ka ethanol a me ka ether solvent, hiki ʻole ke hoʻoheheʻe ʻia i ka wai, hiki ʻole ke hoʻoheheʻe ʻia i loko o ka waikawa hydrochloric dilute, hiki ke hoʻoheheʻe iki ʻia i loko o ka alkali dilute. a i ʻole ka pauka keʻokeʻo ʻē. Ma muli o ke ʻano i hoʻopili ʻia, hiki ʻole ke hoʻoheheʻe ʻia i ka wai; pehu ia ke omo i ka wai.
Hoʻohana: mea hoʻoheheʻe papa, mea hoʻopaʻa, mea hoʻoheheʻe.
3. Methylcellulose (MC):
ʻAno: methyl ether o ka cellulose
Nā Waiwai: Pauka keʻokeʻo a melemele paha a i ʻole nā granules. ʻAʻole hiki ke hoʻoheheʻe ʻia i ka wai wela, ka wai paʻakai momona, ka waiʻona, ka ether, ka acetone, toluene, ka chloroform; hiki ke hoʻoheheʻe ʻia i loko o ka waikawa acetic glacial a i ʻole kahi hui like o ka waiʻona a me ka chloroform. Pili ka solubility i ka wai anuanu i ke kekelē o ka pani ʻana, a ʻoi aku ka maikaʻi o ka hoʻoheheʻe ʻia ʻana i ka wā he 2 ke kekelē o ka pani ʻana.
Hoʻohana: mea hoʻopaʻa papa, matrix o ka mea hoʻoheheʻe papa a i ʻole ka hoʻomākaukau hoʻokuʻu mau ʻia, kirīmi a gel paha, mea hoʻokuʻu a me ka mea hoʻomānoanoa, uhi papa, mea hoʻopaʻa emulsion.
4. ʻEtila kelulose (EC):
ʻAno: Ethyl ether o ka cellulose
Nā Waiwai: Pauka keʻokeʻo a melemele paha a me nā granules. ʻAʻole hiki ke hoʻoheheʻe ʻia i ka wai, nā wai gastrointestinal, glycerol a me propylene glycol. He maʻalahi ka hoʻoheheʻe ʻia i loko o ka chloroform a me ka toluene, a hana i kahi precipitate keʻokeʻo i ka hihia o ka ethanol.
Hoʻohana: He mea lawe wai-hoʻoheheʻe kūpono, kūpono e like me ka matrix lāʻau lapaʻau wai-koʻikoʻi, mea lawe wai-hoʻoheheʻe, mea hoʻopaʻa papa, mea kiʻiʻoniʻoni, mea microcapsule a me ka mea uhi hoʻokuʻu mau, a pēlā aku.
5. Hydroxyethyl Cellulose (HEC):
ʻAno: ʻĀpana hydroxyethyl ether o ka cellulose.
Nā Waiwai: Pauka melemele māmā a keʻokeʻo waiū paha. Hoʻoheheʻe piha ʻia i ka wai anuanu, ka wai wela, ka waikawa nāwaliwali, ke kumu nāwaliwali, ka waikawa ikaika, ke kumu ikaika, ʻaʻole hoʻoheheʻe ʻia i ka hapa nui o nā mea hoʻoheheʻe organik (hoʻoheheʻe ʻia i ka dimethyl sulfoxide, dimethylformamide), i loko o nā mea hoʻoheheʻe organik diol polar Hiki ke hoʻonui a hoʻoheheʻe hapa ʻia paha.
Nā noi: Nā mea polymer wai-soluble non-ionic; nā mea hoʻomānoanoa no nā hoʻomākaukau ophthalmic, otology a me ka hoʻohana topical; HEC i nā lubricants no nā maka maloʻo, nā aniani hoʻopili a me ka waha maloʻo; hoʻohana ʻia i nā mea hoʻonani. Ma ke ʻano he mea hoʻopaʻa, mea hana kiʻiʻoniʻoni, mea hoʻomānoanoa, mea hoʻomaha a me ka mea hoʻopaʻa no nā lāʻau lapaʻau a me ka meaʻai, hiki iā ia ke hoʻopuni i nā ʻāpana lāʻau lapaʻau, i hiki i nā ʻāpana lāʻau lapaʻau ke pāʻani i kahi hana hoʻokuʻu lohi.
6. Hydroxypropyl Cellulose (HPC):
ʻAno: ʻĀpana polyhydroxypropyl ether o ka cellulose
Nā Waiwai: ʻO ka HPC i hoʻololi ʻia he pauka keʻokeʻo a melemele iki paha. Hoʻoheheʻe ʻia i loko o ka methanol, ethanol, propylene glycol, isopropanol, dimethyl sulfoxide a me dimethyl formamide, ʻoi aku ka liʻiliʻi o ka hoʻoheheʻe ʻia o ka viscosity kiʻekiʻe. ʻAʻole hoʻoheheʻe ʻia i ka wai wela, akā hiki ke pehu. Gelation Thermal: maʻalahi ka hoʻoheheʻe ʻia i ka wai ma lalo o 38°C, gelatinized ma ka hoʻomehana ʻana, a hana i ka pehu flocculent ma 40-45°C, hiki ke hoʻihoʻi ʻia ma ka hoʻomaʻalili ʻana.
Nā hiʻohiʻona koʻikoʻi o L-HPC: hiki ʻole ke hoʻoheheʻe ʻia i ka wai a me nā mea hoʻoheheʻe organik, akā hiki ke pehu i ka wai, a piʻi ka waiwai pehu me ka hoʻonui ʻia o nā mea pani
Noi: Hoʻohana ʻia ka HPC i hoʻololi ʻia me he mea hoʻopaʻa papa lāʻau, mea hoʻopili granulating, mea uhi kiʻiʻoniʻoni, a hiki ke hoʻohana ʻia me he mea kiʻiʻoniʻoni microencapsulated, mea matrix a me nā mea kōkua o ka papa paʻa gastric, thickener a me nā colloids pale, i hoʻohana pinepine ʻia i nā ʻāpana transdermal.
L-HPC: Hoʻohana nui ʻia ma ke ʻano he mea hoʻoheheʻe papa a i ʻole he mea hoʻopaʻa no ka granulation pulu, ma ke ʻano he matrix papa hoʻokuʻu mau ʻia, a pēlā aku.
7. Hypromellose (HPMC):
ʻAno: ʻĀpana methyl a me kahi ʻāpana polyhydroxypropyl ether o ka cellulose
Nā Waiwai: Pauka fibrous a granular keʻokeʻo a keʻokeʻo paha. Hiki ke hoʻoheheʻe ʻia i ka wai anuanu, ʻaʻole hiki ke hoʻoheheʻe ʻia i ka wai wela, a he mau waiwai gelation thermal. Hiki ke hoʻoheheʻe ʻia i loko o nā hopena methanol a me ethanol, nā hydrocarbons chlorinated, acetone, a pēlā aku. ʻOi aku ka maikaʻi o kona solubility i nā solvents organik ma mua o ka wai-hoʻoheheʻe ʻia.
Hoʻohana: ʻO kēia huahana he hopena wai haʻahaʻa viscosity i hoʻohana ʻia ma ke ʻano he mea uhi kiʻiʻoniʻoni; hoʻohana ʻia kahi hopena hoʻoheheʻe organik kiʻekiʻe-viscosity e like me kahi mea hoʻopaʻa papa, a hiki ke hoʻohana ʻia ka huahana viscosity kiʻekiʻe e ālai i ka matrix hoʻokuʻu o nā lāʻau lapaʻau wai-hoʻoheheʻe ʻia; e like me ka mea hoʻomānoanoa o nā kulu maka no ka lacquer a me nā waimaka artificial, a me ka mea hoʻomaʻū no nā aniani hoʻopili.
8. Hypromellose Phthalate (HPMCP):
ʻAno: ʻO HPMCP ka hapalua ester waikawa phthalic o HPMC.
Nā Waiwai: Nā ʻāpana beige a keʻokeʻo paha a i ʻole nā granules. ʻAʻole hiki ke hoʻoheheʻe ʻia i ka wai a me ka hopena waikawa, ʻaʻole hiki ke hoʻoheheʻe ʻia i ka hexane, akā maʻalahi ka hoʻoheheʻe ʻia i ka acetone:methanol, acetone:ethanol a i ʻole methanol:chloromethane.
Noi: He ʻano mea uhi hou me ka hana maikaʻi loa, hiki ke hoʻohana ʻia e like me ka uhi ʻiliʻili e uhi i ke ʻala ʻano ʻē o nā papa a i ʻole nā granules.
9. Hypromellose Acetate Succinate (HPMCAS):
ʻAno: Nā esters acetic a me succinic i hui pū ʻia oHPMC
Nā Waiwai: Pauka keʻokeʻo a melemele paha a i ʻole nā granules. Hoʻoheheʻe ʻia i loko o ka sodium hydroxide a me ka sodium carbonate solution, maʻalahi ka hoʻoheheʻe ʻia i loko o ka acetone, methanol a i ʻole ethanol: wai, dichloromethane: hui ethanol, ʻaʻole hoʻoheheʻe ʻia i ka wai, ethanol a me ether.
Hoʻohana: Ma ke ʻano he mea uhi enteric papa, mea uhi hoʻokuʻu mau a me nā mea uhi kiʻiʻoniʻoni.
10. ʻAka:
ʻAno: ʻO Agar kahi hui ʻana o ʻelua mau polysaccharides ma ka liʻiliʻi, ma kahi o 60-80% agarose kūlike a me 20-40% agarose. Ua haku ʻia ʻo Agarose me nā ʻāpana e hana hou ana i ka agarobiose kahi i hoʻopili ʻokoʻa ʻia ai ʻo D-galactopyranosose a me L-galactopyranosose ma 1-3 a me 1-4.
Nā Waiwai: He ʻano translucent ʻo Agar, he melemele māmā kona ʻano, he ʻāpana lahilahi a unahi paha a he pauka paha. ʻAʻole hoʻoheheʻe ʻia i ka wai anuanu, hoʻoheheʻe ʻia i ka wai e paila ana. Hoʻonui ʻia i 20 mau manawa i ka wai anuanu.
Hoʻohana: Ma ke ʻano he mea hoʻopaʻa, kumu poni, kumu suppository, emulsifier, stabilizer, suspending agent, e like me ka poultice, capsule, syrup, jelly a me ka emulsion.
Ka manawa hoʻouna: ʻApelila-26-2024