1. Sodium ya Croscarmellose(guhuza CMCNa): guhuza cololymer ya CMCNa
Ibyiza: Ifu yera cyangwa itari yera. Bitewe nuburyo buhujwe, ntibishobora gushonga mumazi; irabyimba vuba mumazi kugeza inshuro 4-8 ubwinshi bwumwimerere. Ifu ifite amazi meza.
Porogaramu: Nibisanzwe bikoreshwa cyane super disintegrant. Gutandukana kumunwa wibinini, capsules, granules.
2. Kalisiyumu ya Carmellose (ihuza CMCCa):
Ibyiza: Ifu yera, impumuro nziza, hygroscopique. 1% igisubizo pH 4.5-6. Hafi ya elegitoronike muri Ethanol na ether solvent, idashonga mumazi, idashobora gushonga muri acide hydrochloric acide, gushonga gake muri alkali. cyangwa ifu yera. Bitewe nuburyo buhujwe, ntibishobora gushonga mumazi; irabyimba iyo ikurura amazi.
Porogaramu: tablet disintegrant, binder, diluent.
3. Methylcellulose (MC):
Imiterere: methyl ether ya selile
Ibyiza: Ifu yera cyangwa umuhondo ifu yera cyangwa granules. Kudashonga mumazi ashyushye, umunyu wuzuye, inzoga, ether, acetone, toluene, chloroform; gushonga muri acide acetike glacial cyangwa imvange ingana ya alcool na chloroform. Gukomera mumazi akonje bifitanye isano nurwego rwo gusimburwa, kandi birashobora gukemuka cyane iyo urwego rwo gusimburwa ari 2.
Gushyira mu bikorwa: ibinini bya tableti, matrix ya tablet isenya ibintu cyangwa gutegura-kurekura-gusohora, cream cyangwa gel, guhagarika ibintu hamwe no kubyimba, ibinini bya tableti, stabilisateur ya emulsion.
4. Ethyl selulose (EC):
Imiterere: Ethyl ether ya selile
Ibyiza: Ifu yera cyangwa umuhondo-yera ifu na granules. Kudashonga mumazi, gastrointestinal fluid, glycerol na propylene glycol. Irashobora gushonga byoroshye muri chloroform na toluene, kandi ikora imvura yera mugihe habaye Ethanol.
Gushyira mu bikorwa: Ikintu cyiza cyogutwara amazi adashobora gushonga, gikwiye nka matrike yibiyobyabwenge byamazi, itwara amazi adashobora gushonga, ibinini bya tableti, ibikoresho bya firime, ibikoresho bya microcapsule hamwe nibikoresho byo gutwikira bikomeza, nibindi.
5. Hydroxyethyl Cellulose (HEC):
Imiterere: Hydroxyethyl igice cya selile.
Ibyiza: Ifu yera yumuhondo cyangwa amata. Kurandura byuzuye mumazi akonje, amazi ashyushye, acide idakomeye, ishingiro ridakomeye, acide ikomeye, base ikomeye, idashobora gushonga mumashanyarazi menshi (gushonga muri dimethyl sulfoxide, dimethylformamide), mumashanyarazi ya diol polar irashobora kwaguka cyangwa gushonga igice.
Gusaba: Ibikoresho bitari ionic amazi-soluble ibikoresho bya polymer; umubyimba wo gutegura amaso, otologiya no gukoresha ibintu; HEC mumavuta yo kwisiga amaso yumye, guhuza imiyoboro hamwe numunwa wumye; ikoreshwa mu kwisiga. Nkumuhuza, ukora firime, umubyimba, guhagarika imiti hamwe na stabilisateur kumiti nibiryo, irashobora gukwirakwiza ibice byibiyobyabwenge, kugirango ibice byibiyobyabwenge bigire uruhare mukurekura buhoro.
6. Hydroxypropyl Cellulose (HPC):
Imiterere: Igice cya polyhydroxypropyl ether ya selile
Ibyiza: HPC isimbuwe cyane ni ifu yera cyangwa ifu yumuhondo. Gukemuka muri methanol, Ethanol, propylene glycol, isopropanol, dimethyl sulfoxide na formetide ya dimethyl, verisiyo yo hejuru ya viscosity ntishobora gukemuka. Kudashonga mumazi ashyushye, ariko birashobora kubyimba. Ubushyuhe bwa Thermal: gushonga byoroshye mumazi ari munsi ya 38 ° C, gelatine ukoresheje ubushyuhe, kandi bigatera kubyimba flokculent kuri 40-45 ° C, bishobora kugarurwa no gukonjesha.
L-HPC ibintu byingenzi biranga: kudashonga mumazi no mumashanyarazi, ariko kubyimba mumazi, kandi imitungo yabyimbye yiyongera hamwe no kwiyongera kwinsimburangingo.
Gushyira mu bikorwa: HPC isimbuwe cyane ikoreshwa nka tablet binder, agent granulation agent, material coating material, kandi irashobora kandi gukoreshwa nkibikoresho bya firime ya microencapsulée, ibikoresho bya matrix nibikoresho bifasha ibikoresho byo kugaburira gastrica, kubyimbye hamwe na Protective colloids, nabyo bikunze gukoreshwa muburyo bwa transdermal.
L-HPC.
7. Hypromellose (HPMC):
Imiterere: Methyl igice hamwe na polyhydroxypropyl ether ya selile
Ibyiza: Fibrous yera cyangwa yera-ifu cyangwa ifu ya granular. Irashobora gushonga mumazi akonje, idashonga mumazi ashyushye, kandi ifite imiterere yubushyuhe. Irashobora gushonga muri methanol na Ethanol ibisubizo, hydrocarbone ya chlorine, acetone, nibindi.
Gushyira mu bikorwa: Iki gicuruzwa nigisubizo gito cyamazi yo mumazi akoreshwa nkibikoresho bya firime; igisubizo cyinshi-cyinshi cyibisubizo byumuti bikoreshwa nkibikoresho bya tablet, kandi ibicuruzwa byinshi-viscosity birashobora gukoreshwa muguhagarika matrix irekura imiti ibora amazi; nkuko ijisho ritonyanga cyane kuri lacquer n'amarira yubukorikori, hamwe nogukoresha ibikoresho byo guhuza.
8. Hypromellose Phthalate (HPMCP):
Imiterere: HPMCP ni acide phthalic igice cya ester ya HPMC.
Ibyiza: Beige cyangwa flake yera cyangwa granules. Kudashonga mumazi nigisubizo cya acide, ntigishobora gushonga muri hexane, ariko byoroshye gushonga muri acetone: methanol, acetone: Ethanol cyangwa methanol: ivangwa rya chloromethane.
Gushyira mu bikorwa: Ubwoko bushya bwibikoresho bifatika hamwe nibikorwa byiza, bishobora gukoreshwa nka firime ya firime kugirango uhishe impumuro idasanzwe yibinini cyangwa granules.
9. Hypromellose Acetate Succinate (HPMCAS):
Imiterere: Imvange ya acetike na succinic esters yaHPMC
Ibyiza: Ifu yera cyangwa umuhondo ifu yera cyangwa granules. Gushonga muri sodium hydroxide na sodium ya karubone yumuti, byoroshye gushonga muri acetone, methanol cyangwa Ethanol: amazi, dichloromethane: imvange ya Ethanol, idashonga mumazi, Ethanol na ether.
Gushyira mu bikorwa: Nka tablet enteric coating material, ibikoresho byo gusohora bikomeza hamwe nibikoresho bya firime.
10. Agar:
Imiterere: Agar ni imvange byibura polysaccharide ebyiri, hafi 60-80% agarose idafite aho ibogamiye na agarose 20-40%. Agarose igizwe na agarobiose isubiramo ibice aho D-galactopyranosose na L-galactopyranosose bisimburana kuri 1-3 na 1-4.
Ibyiza: Agar irasobanutse, silindari yumuhondo yoroheje yumuhondo, umurongo woroshye cyangwa flake flake cyangwa ibintu byifu. Kudashonga mumazi akonje, gushonga mumazi abira. Kubyimba inshuro 20 mumazi akonje.
Gusaba: Nka agent ihuza, amavuta yo kwisiga, base suppository, emulsifier, stabilisateur, agent uhagarika, nanone nka poultice, capsule, sirupe, jelly na emulsion.
Igihe cyo kohereza: Apr-26-2024